Activella 1 mg-0.5 mg tablet is a prescription Hormone Replacement Therapy (HRT) mainly used to overcome menopausal symptoms in women, including hot flashes and mood swings. It includes two FDA-approved active ingredients, 1 mg estradiol (an estrogen) and 0.5 mg norethindrone acetate (a progestin).
It belongs to the estrogen-progestin combination class, manufactured by Novo Nordisk in a GMP-compliant facility. Estradiol restores diminishing estrogen levels, reducing hot flashes and vaginal shrinkage. On the other hand, norethindrone protects the uterus by reducing the risk of endometrial (the inner lining of the uterus) overgrowth caused by estrogen alone.
Activella is mainly used to manage moderate to severe menopausal symptoms and to help prevent postmenopausal Osteoporosis in women at risk when other treatments are unsuitable.
The usual prescribed dose is one pill a day taken at the same time every day. If you miss a dosage, have it as soon as you recall. However, if it is nearly time for your next dose, ignore your missed dose and continue with your regular schedule.
An overdose can induce nausea or breast soreness, requiring immediate medical attention. Common adverse effects include breast discomfort, headaches, nausea, and irregular vaginal bleeding. If you experience any symptoms of blood clots, chest discomfort, or unexpected eyesight changes, obtain medical help immediately.
Do not use if you have a history of undiagnosed vaginal bleeding, Breast Cancer, or blood clots. Keep the medication at room temperature, away from heat, moisture, and direct sunlight.
Activella works by combining estradiol and norethindrone acetate to help postmenopausal women regain hormonal balance. Estradiol replaces declining estrogen levels, helping maintain vaginal and bone health. Norethindrone acetate, a progestin, reduces the impact of estrogen on the uterus, lowering the risk of endometrial thickening. Its main benefits include:
Always follow your doctor's instructions to ensure the best results and safety when using this menopause tablet. A few general usage guidelines are:
Currently, there are no other strengths available for this menopause symptom relief tablet at Cheap Medicine Shop. If you are looking for any other strengths, explore the following alternatives after consulting your medical provider:
| Estrabet 2 Tablet | $6.00/ 10 pills |
| Evatone 2 Tablet | $3.80/ 10 pills |
Activella tablet commonly causes mild effects like:
These effects are often temporary and improve over time as your body adjusts to the medication. In case they persist or turn bothersome, reach out to your medical provider immediately.
Liver Disease
Patients with liver disease should avoid taking Activella tablets since hormone treatment can affect liver function. It should only be taken if specifically recommended by a doctor after a thorough examination and regular liver monitoring.
Kidney Impairment
Kidney patients should exercise caution when taking Activella since hormone treatment can cause fluid retention and electrolyte imbalance, which can affect kidney function. Decreased kidney function can also reduce medication clearance from the body, raising the likelihood of unwanted effects. Hence, frequent monitoring and medical guidance are required.
Pregnant and Breastfeeding women
Activella tablets should not be taken when pregnant or breastfeeding. It could harm the unborn child and be transferred into breast milk, thus affecting milk supply and the breastfeeding newborn.
Avoid
Avoid excess alcohol intake while taking Activella, as it can increase side effects like dizziness, nausea, or liver strain.
Yes, Activella can cause slight weight fluctuations in some women, primarily because of fluid retention or hormonal effects. Significant weight gain is uncommon. A balanced diet, regular exercise, and a healthy lifestyle can help you manage your weight during treatment.
Activella usually starts relieving menopausal symptoms like hot flashes and night sweats within 1–2 weeks. However, complete benefits, especially for bone protection, can take several weeks to a few months of regular use.
The best time to take Activella is once a day at the same time, preferably in the morning or evening, whichever suits your routine. Consistent use helps to maintain stable hormone levels and enhances treatment efficacy.
Activella is a continuous hormone treatment; therefore, you will not experience regular menstrual periods while taking it. However, minor spotting or sudden bleeding can occur, particularly in the first few months of treatment.
The use of Activella should only be done after a doctor's approval. It could be discontinued if menopausal symptoms resolve, side effects become severe, or conditions like blood clots, Breast Cancer, liver problems, or unexplained vaginal bleeding develop.
Yes, Activella can sometimes cause High Blood Pressure due to its estrogen content. Hence, regular monitoring is required. Also, consult your doctor if you notice persistent increases or related symptoms.
Yes, Activella can cause hair loss in some women, though it is uncommon. Hormonal changes from estrogen–progestin therapy can affect hair growth. If hair thinning persists or is severe, consult your doctor.
