ana@cheapmedicineshop.com
Store Phone Numbers 
Telegram
Anestol Ointment 5% (30 gm)
Offer You Can't Resist
Free Shipping
What is Anestol Ointment 5%
Anestol Ointment 5% is formulated with EMA (European Medicines Agency) and FDA-approved Lidocaine to temporarily block nerve signals in the skin. By stabilizing neuronal membranes, it reduces pain sensations at the site of application. This prescription-strength topical skin numbing cream is manufactured by GMP-compliant Sandoz Pharma.
Lidocaine belongs to the chemical class acetamide, 2-(diethylamino)-N - (2,6-dimethylphenyl) and is categorized as a local anesthetic and antiarrhythmic agent. It is sold under brand names, such as Anestol, Xylocaine, Aspercreme, Topicaine, Burnamycin and Solarcaine First Aid, in the USA and Canada.
Topical lidocaine solutions have a rapid onset on mucosal or compromised skin. They are widely used for relief from Localized Neuropathic Pain (LNP), minor burn treatment, skin irritation, hemorrhoid-associated discomfort, and injection-site numbing.
Patients may temporarily feel nausea, headache or dizziness, while excessive or frequent use may cause serious cardiovascular or nervous system damage. Moreover, it should be used cautiously in children and the elderly due to the risk of greater skin permeability and comorbidities, respectively. So, make sure to inform your doctor of your age and medications/supplements you are taking currently to avoid serious drug interactions.
What are the benefits of taking Anestol Ointment 5%
Lidocaine acts by blocking sodium channels on nerve endings. This temporarily halts pain signal transmission, creating a numbing effect at the area of application. Anestol uses and benefits include:
- Fast local numbing: Onset occurs within 3 to 5 minutes.
- Long-lasting relief: Its numbing effect can last for up to 1-2 hours.
- Focused action: It acts at the skin/nerve endings with minimal systemic exposure when used as directed.
- Procedural comfort: Clinical studies show that 5% Lidocaine ointment reduces pain severity during skin injections and routine minor procedures. Moreover, it helps with anxiety-related discomfort around minor procedures.
How to take Anestol Ointment 5%
Make sure to learn about proper dosage and use from your doctor to limit systemic absorption and side effects. Then, follow the given steps to safely use Anestol cream, gel or ointment:
- Wash your hands and the affected area before application.
- Apply a thin layer to the affected, unbroken skin as directed by your clinician.
- Do not apply heat or heating pads.
- Avoid tight dressings over the application site.
- Wash your hands after use and avoid touching your eyes, nose or mouth.
- Use only on the outside of the body and do not use inside body cavities unless directed.
- If using for hemorrhoid pain or anal fissures, apply as instructed after bowel movements.
- Do not use more than recommended or on other areas, as it may increase systemic absorption.
Store it at room temperature between 68° and 77°F (20-25°C) in a dry area away from sunlight. Keep all topical anesthetics out of reach of children and pets, as accidental ingestion or excessive exposure can be dangerous and require emergency medical care.
Anestol ointment dosage varies by age group and condition being treated. Typical recommendations are as follows:
- For Adults: Apply a small amount up to 5g per use; no more than 20g per day. It is usually applied 2-3 times daily, depending on the severity of your condition and location.
- For children: Your pediatrician will adjust the dosage to a maximum of 4.5 mg/kg or 2 mg/lb.
Strengths and Substitutes
Anestol ointment is currently available in a 5% Lidocaine 30 mg tube for topical use. Lidocaine formulations, however, also exist as gels, sprays, medicated patches for nerve pain relief and topical dental anesthetics.
You can explore other substitutes at 50-80% lower rates at Cheap Medicine Shop.
| $1.46/ tube | |
| $8.96/ tube |
What are the side effects of Anestol
Adverse reactions with topical Lidocaine 5% are mostly mild, local and application-site related. Common side effects of Anestol include:
- Headache
- Unusual weakness or fatigue
- Nausea or vomiting
- Lightheadedness or dizziness
- Shortness of breath
- Allergic reactions like skin rash, hives or facial swelling
Most of these are temporary; however, seek medical advice if symptoms persist or severe effects like allergic reactions, cardiovascular effects, or respiratory depression are observed.
Safety advice
Liver disease
Discuss dosing limits with your clinician and use cautiously, as it may raise systemic levels.
Kidney impairment
Elderly patients should only use Anestol under medical advice due to skin permeability and comorbidity risks.
Pregnant and breastfeeding women
Topical use of Lidocaine may be permissible under medical supervision, but confirm risks and benefits with a clinician before use. Avoid large areas and prolonged exposure.
Due to greater skin permeability in kids, higher vigilance is needed with children.
Avoid
Do not apply to broken/irritated skin and avoid large areas to prevent excessive absorption and toxicity.
Certain medicines (beta-blockers, class I antiarrhythmics) may increase cardiac or CNS effects. Inform your doctor about all prescription and non-prescription medicines, as well as supplements and existing health conditions.
Do not use if you’ve had hypersensitivity to amide-type local anesthetics. Seek immediate care if swelling, wheeze, or severe rash occurs.
FAQs
Does Lidocaine speed up healing?
No, Lidocaine is a numbing agent that reduces pain signals but does not accelerate tissue repair. It can make daily care more comfortable, which might help you tolerate wound cleaning or minor procedures. Still, healing will depend on the underlying cause and appropriate medical care.
Can you still feel pain with Lidocaine?
Yes, it is possible. Topical Lidocaine dulls pain and itch but may not completely block pressure or deep pain. Pain relief depends on ointment dosage, frequency, contact time, and the thickness of the skin where it is applied.
Is Lidocaine cream a steroid?
No, Lidocaine is a local anesthetic, not a corticosteroid. It numbs nerve endings to reduce localised pain and itch. Steroid creams, on the other hand, reduce inflammation.
Can you buy Lidocaine 5% ointment over the counter?
Yes, some lower-strength products are OTC (over-the-counter), while 5% topical Anestol ointments or creams may require a prescription. Ask your pharmacist or clinician about local regulations, as Lidocaine availability varies by country and formulation.
How long does Lidocaine ointment take to work?
Numbing typically begins within a few minutes on suitable application sites, depending on skin condition and thickness. However, Anestol use on intact skin may have a slower or more limited effect.
How long does Lidocaine last for pain relief?
The duration of treatment depends on the dose and frequency prescribed, application site, and whether the skin is intact at the site. Anestol pain relief often persists for short intervals and is suitable for minor procedures or localized pain flares. Make sure to reapply only as directed, as excessive frequency or amount increases systemic risk.
Is Lidocaine 5% safe to use?
Yes, 5% topical Lidocaine is generally safe and well-tolerated when used as directed on small areas of unbroken skin. However, overuse leading to blockage, or application to large/broken areas, can raise blood levels and cause serious side effects.
Is Anestol used for sunburn?
Yes, topical Lidocaine or Anestol can ease sunburn-related pain, itch and even mosquito/bug bite pain, but it should be used sparingly. Seek medical care for extensive burns, blistering, or signs of infection.
What happens if you use too much Lidocaine 5%?
Overuse or application to large/broken areas can cause excessive Lidocaine absorption, leading to seizures, irregular heartbeat, chest pain, or breathing problems. It can also cause Methemoglobinemia, a rare but serious condition in which haemoglobin is altered so it cannot carry oxygen effectively. Symptoms include gray or bluish lips and skin, headache, dizziness, shortness of breath, and fatigue.
What happens if Lidocaine hits a nerve?
Topical ointment like Lidocaine acts on surface nerve endings and is not injected. Thus, excessive absorption, use on broken skin or use for teething pain can produce CNS or cardiovascular symptoms such as dizziness, confusion or arrhythmias.
Who should not use Lidocaine ointment?
You should not use Lidocaine if you’ve had amide-type anesthetic allergy, significant liver dysfunction or renal issues. Since this medication crosses the placenta and is excreted into breast milk, it should only be used by pregnant or breastfeeding women under medical supervision.